CU-CPT8m [Ligand Id: 9795] activity data from GtoPdb

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  • TLR8 in Human [GtoPdb: 1758] [UniProtKB: Q9NR97]
Created with Highcharts 10.3.3ValuesChart context menuTLR8pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TLR8 in Human [GtoPdb: 1758] [UniProtKB: Q9NR97]
GtoPdb Dissociation constant measured using isothermal titration calorimetry (ITC) and the hTRL8 ectodomain. - 6.66 pKd 220 nM Kd Nat Chem Biol (2018) 14: 58-64 [PMID:29155428]
GtoPdb - - 7.17 pIC50 67 nM IC50 Nat Chem Biol (2018) 14: 58-64 [PMID:29155428]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.