rogaratinib [Ligand Id: 9789] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362] | ||||||||
| GtoPdb | At a high ATP level. | - | 7.91 | pKi | 12.2 | nM | Ki | WO2013087578. Disubstituted benzothienyl-pyrrolotriazines and their use as FGFR kinase inhibitors (2013) |
| fibroblast growth factor receptor 3 in Human [GtoPdb: 1810] [UniProtKB: P22607] | ||||||||
| GtoPdb | - | - | 7.61 | pIC50 | 24.8 | nM | IC50 | WO2013087578. Disubstituted benzothienyl-pyrrolotriazines and their use as FGFR kinase inhibitors (2013) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
