PBT-3 [Ligand Id: 9755] activity data from GtoPdb

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  • TP receptor in Human [GtoPdb: 346] [UniProtKB: P21731]
Created with Highcharts 10.3.3ValuesChart context menuTP receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TP receptor in Human [GtoPdb: 346] [UniProtKB: P21731]
GtoPdb Antagonism of TPbeta (long) isoform expressed in COS7 cells. - 5.92 pIC50 1200 nM IC50 J Pharmacol Exp Ther (2003) 307: 1142-7 [PMID:14560042]
GtoPdb Antagonism of TPalpha (short) isoform expressed in COS7 cells. - 6.7 pIC50 200 nM IC50 J Pharmacol Exp Ther (2003) 307: 1142-7 [PMID:14560042]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.