semaglutide [Ligand Id: 9724] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GLP-1 receptor in Human [GtoPdb: 249] [UniProtKB: P43220] | ||||||||
| GtoPdb | Membrane radioligand displacement assay (125I-GLP-1 as tracer) performed in the absence of human serum albumin. | - | 9.42 | pIC50 | 0.38 | nM | IC50 | J Med Chem (2015) 58: 7370-80 [PMID:26308095] |
| GtoPdb | In vitro potency assessed in BHK cells expressing the human GLP-1R and a luciferase reporter system. | - | 11.21 | pEC50 | 0.01 | nM | EC50 | J Med Chem (2015) 58: 7370-80 [PMID:26308095] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
