compound 5e [PMID: 28580438] [Ligand Id: 9712] activity data from GtoPdb

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  • platelet derived growth factor receptor beta in Human [GtoPdb: 1804] [UniProtKB: P09619]
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  • fms related receptor tyrosine kinase 3 in Human [GtoPdb: 1807] [UniProtKB: P36888]
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  • Janus kinase 1 in Human [GtoPdb: 2047] [UniProtKB: P23458]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
platelet derived growth factor receptor beta in Human [GtoPdb: 1804] [UniProtKB: P09619]
GtoPdb - - 7.55 pKd 28 nM Kd ACS Omega (2017) 2: 1985-2009 [PMID:28580438]
fms related receptor tyrosine kinase 3 in Human [GtoPdb: 1807] [UniProtKB: P36888]
GtoPdb Measured using the Z′-LYTE Kinase Assay Kit and wild type FLT3. - 8.44 pKd 3.6 nM Kd ACS Omega (2017) 2: 1985-2009 [PMID:28580438]
Janus kinase 1 in Human [GtoPdb: 2047] [UniProtKB: P23458]
GtoPdb Measured using the JAK1 JH2 domain-pseudokinase. - 7.55 pKd 28 nM Kd ACS Omega (2017) 2: 1985-2009 [PMID:28580438]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.