Takinib [Ligand Id: 9655] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CDC like kinase 2 in Human [GtoPdb: 1991] [UniProtKB: P49760] | ||||||||
| GtoPdb | - | - | 6.37 | pIC50 | 430 | nM | IC50 | Cell Chem Biol (2017) 24: 1029-1039.e7 [PMID:28820959] |
| interleukin 1 receptor associated kinase 1 in Human [GtoPdb: 2042] [UniProtKB: P51617] | ||||||||
| GtoPdb | - | - | 6.41 | pIC50 | 390 | nM | IC50 | Cell Chem Biol (2017) 24: 1029-1039.e7 [PMID:28820959] |
| interleukin 1 receptor associated kinase 4 in Human [GtoPdb: 2045] [UniProtKB: Q9NWZ3] | ||||||||
| GtoPdb | - | - | 6.92 | pIC50 | 120 | nM | IC50 | Cell Chem Biol (2017) 24: 1029-1039.e7 [PMID:28820959] |
| mitogen-activated protein kinase kinase kinase 7 in Human [GtoPdb: 2082] [UniProtKB: O43318] | ||||||||
| GtoPdb | In vitro kinase activity assay, measuring phosphorylation of a peptide substrate by a purified recombinant TAK1 kinase domain fused to TAB1 c-terminal domain. | - | 8.02 | pIC50 | 9.5 | nM | IC50 | Cell Chem Biol (2017) 24: 1029-1039.e7 [PMID:28820959] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
