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ChEMBL ligand: CHEMBL3707398 (Asivatrep, Pac-14028) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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TRPV1 in Rat [GtoPdb: 507] [UniProtKB: O35433] | ||||||||
GtoPdb | Antagonism of capsaicin-induced calcium influx in isolated primary rat spinal dorsal root ganglia cells. | - | 8.21 | pIC50 | 6.2 | nM | IC50 | US7858621. Compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist; and pharmaceutical compositions containing the same (2010) |
ChEMBL data shown on this page come from version 31:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]