BMS-202 [Ligand Id: 9607] activity data from GtoPdb

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  • CB1 receptor in Human [GtoPdb: 56] [UniProtKB: P21554]
Created with Highcharts 10.3.3ValuesChart context menuCB1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • CB2 receptor in Human [GtoPdb: 57] [UniProtKB: P34972]
Created with Highcharts 10.3.3ValuesChart context menuCB2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CB1 receptor in Human [GtoPdb: 56] [UniProtKB: P21554]
GtoPdb - - 6.99 pIC50 102 nM IC50 ACS Chem Neurosci (2015) 6: 1445-58 [PMID:25921407]
CB2 receptor in Human [GtoPdb: 57] [UniProtKB: P34972]
GtoPdb - - 6.88 pEC50 131 nM EC50 ACS Chem Neurosci (2015) 6: 1445-58 [PMID:25921407]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.