C391 [Ligand Id: 9570] activity data from GtoPdb

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  • PAR2 in Human [GtoPdb: 348] [UniProtKB: P55085]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
PAR2 in Human [GtoPdb: 348] [UniProtKB: P55085]
GtoPdb Antagonism of 2-at-LIGRL-NH2-induced ERK phosphorylation in 16HBE14o- cells. - 4.84 pIC50 14300 nM IC50 Br J Pharmacol (2015) 172: 4535-4545 [PMID:26140338]
GtoPdb Antagonism of peptidomimetic-induced PAR2 Ca2+ signalling in 16HBE14o- cells. - 5.89 pIC50 1300 nM IC50 Br J Pharmacol (2015) 172: 4535-4545 [PMID:26140338]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.