C391 [Ligand Id: 9570] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| PAR2 in Human [GtoPdb: 348] [UniProtKB: P55085] | ||||||||
| GtoPdb | Antagonism of 2-at-LIGRL-NH2-induced ERK phosphorylation in 16HBE14o- cells. | - | 4.84 | pIC50 | 14300 | nM | IC50 | Br J Pharmacol (2015) 172: 4535-4545 [PMID:26140338] |
| GtoPdb | Antagonism of peptidomimetic-induced PAR2 Ca2+ signalling in 16HBE14o- cells. | - | 5.89 | pIC50 | 1300 | nM | IC50 | Br J Pharmacol (2015) 172: 4535-4545 [PMID:26140338] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
