MS049 [Ligand Id: 9529] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| coactivator associated arginine methyltransferase 1 in Human [GtoPdb: 1255] [UniProtKB: Q86X55] | ||||||||
| GtoPdb | Isothermal titration calorimetry (ITC) in the presence of SAH | - | 7 | pKd | 100 | nM | Kd | J Med Chem (2016) 59: 9124-9139 [PMID:27584694] |
| GtoPdb | - | - | 7.47 | pIC50 | 34 | nM | IC50 | J Med Chem (2016) 59: 9124-9139 [PMID:27584694] |
| protein arginine methyltransferase 6 in Human [GtoPdb: 1257] [UniProtKB: Q96LA8] | ||||||||
| GtoPdb | Isothermal titration calorimetry (ITC) in the presence of SAH | - | 7.06 | pKd | 87 | nM | Kd | J Med Chem (2016) 59: 9124-9139 [PMID:27584694] |
| GtoPdb | - | - | 7.37 | pIC50 | 43 | nM | IC50 | J Med Chem (2016) 59: 9124-9139 [PMID:27584694] |
| protein arginine methyltransferase 8 in Human [GtoPdb: 1259] [UniProtKB: Q9NR22] | ||||||||
| GtoPdb | - | - | 5.8 | pIC50 | 1600 | nM | IC50 | J Med Chem (2016) 59: 9124-9139 [PMID:27584694] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
