YM-244769 [Ligand Id: 9484] activity data from GtoPdb

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  • Sodium/calcium exchanger 3 in Human [GtoPdb: 947] [UniProtKB: P57103]
Created with Highcharts 10.3.3ValuesChart context menuSodium/calcium exchanger 3pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Sodium/calcium exchanger 3 in Human [GtoPdb: 947] [UniProtKB: P57103]
GtoPdb Inhibition of intracellular Na(+)-dependent [45]Ca(2+) uptake via NCX3. - 7.74 pIC50 18 nM IC50 Mol Pharmacol (2006) 70: 2075-83 [PMID:16973719]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.