CCR2-RA-[R] [Ligand Id: 9431] activity data from GtoPdb

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  • CCR2 in Human [GtoPdb: 59] [UniProtKB: P41597]
Created with Highcharts 10.3.3ValuesChart context menuCCR2pKd HumanpKi HumanpIC50 HumanpEC50 Human0123456Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CCR2 in Human [GtoPdb: 59] [UniProtKB: P41597]
GtoPdb Antagonism of 125I-MCP-1 binding to THP-1 cells - 5.3 pIC50 <5000 nM IC50 Lett Drug Des Discov (2007) 4: 263-271;
US6936633. Pyrrolidinone derivatives (2005)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.