CX-5011 [Ligand Id: 9373] activity data from GtoPdb

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  • Casein kinase 2 in Human [GtoPdb: 1548]
  • Casein kinase 2 in Rat [GtoPdb: 1548]
Created with Highcharts 10.3.3ValuesChart context menuCasein kinase 2pKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
  • Pim-1 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2158] [UniProtKB: P11309]
Created with Highcharts 10.3.3ValuesChart context menuPim-1 proto-oncogene, serine/threonine kinasepKd HumanpKi HumanpIC50 HumanpEC50 Human0123456Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Casein kinase 2 in Human [GtoPdb: 1548]
GtoPdb Recombinant holoenzyme with wild-type alpha subunits. - 8.64 pIC50 2.3 nM IC50 Biochemistry (2011) 50: 8478-88 [PMID:21870818]
Casein kinase 2 in Rat [GtoPdb: 1548]
GtoPdb Native rat CK2 isolated from liver. - 9.01 pIC50 0.97 nM IC50 Biochemistry (2011) 50: 8478-88 [PMID:21870818]
Pim-1 proto-oncogene, serine/threonine kinase in Human [GtoPdb: 2158] [UniProtKB: P11309]
GtoPdb - - 5.6 pIC50 2510 nM IC50 Biochemistry (2011) 50: 8478-88 [PMID:21870818]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.