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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372] | ||||||||
| GtoPdb | - | - | 8.96 | pKi | 1.1 | nM | Ki | Nature (2016) 537: 185-190 [PMID:27533032] |
| GtoPdb | In a Gi/o activation assay. | - | 8.34 | pEC50 | 4.6 | nM | EC50 | Nature (2016) 537: 185-190 [PMID:27533032] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.