adriforant [Ligand Id: 8985] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1915540
  • H3 receptor in Human [GtoPdb: 264] [UniProtKB: Q9Y5N1]
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  • H4 receptor in Human [GtoPdb: 265] [UniProtKB: Q9H3N8]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
H3 receptor in Human [GtoPdb: 264] [UniProtKB: Q9Y5N1]
GtoPdb - - 6.73 pKi - - - Pharmacol. Rev. (2015) 67: 601-55 [PMID:26084539]
H4 receptor in Human [GtoPdb: 265] [UniProtKB: Q9H3N8]
GtoPdb - - 8.31 pKi - - - Pharmacol. Rev. (2015) 67: 601-55 [PMID:26084539]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]