cerdulatinib [Ligand Id: 8957] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| AMP kinase in Human [GtoPdb: 1540] | ||||||||
| GtoPdb | - | - | 8.22 | pIC50 | 6 | nM | IC50 | J Pharmacol Exp Ther (2014) 351: 538-48 [PMID:25253883] |
| colony stimulating factor 1 receptor in Human [GtoPdb: 1806] [UniProtKB: P07333] | ||||||||
| GtoPdb | - | - | 8.3 | pIC50 | 5 | nM | IC50 | J Pharmacol Exp Ther (2014) 351: 538-48 [PMID:25253883] |
| Janus kinase 1 in Human [GtoPdb: 2047] [UniProtKB: P23458] | ||||||||
| GtoPdb | - | - | 7.92 | pIC50 | 12 | nM | IC50 | J Pharmacol Exp Ther (2014) 351: 538-48 [PMID:25253883] |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | - | - | 8.22 | pIC50 | 6 | nM | IC50 | J Pharmacol Exp Ther (2014) 351: 538-48 [PMID:25253883] |
| Janus kinase 3 in Human [GtoPdb: 2049] [UniProtKB: P52333] | ||||||||
| GtoPdb | - | - | 8.1 | pIC50 | 8 | nM | IC50 | J Pharmacol Exp Ther (2014) 351: 538-48 [PMID:25253883] |
| mitogen-activated protein kinase kinase kinase 9 in Human [GtoPdb: 2084] [UniProtKB: P80192] | ||||||||
| GtoPdb | - | - | 8.3 | pIC50 | 5 | nM | IC50 | J Pharmacol Exp Ther (2014) 351: 538-48 [PMID:25253883] |
| NUAK family kinase 1 in Human [GtoPdb: 2129] [UniProtKB: O60285] | ||||||||
| GtoPdb | - | - | 8.4 | pIC50 | 4 | nM | IC50 | J Pharmacol Exp Ther (2014) 351: 538-48 [PMID:25253883] |
| serine/threonine kinase 4 in Human [GtoPdb: 2225] [UniProtKB: Q13043] | ||||||||
| GtoPdb | - | - | 8.4 | pIC50 | 4 | nM | IC50 | J Pharmacol Exp Ther (2014) 351: 538-48 [PMID:25253883] |
| spleen associated tyrosine kinase in Human [GtoPdb: 2230] [UniProtKB: P43405] | ||||||||
| GtoPdb | - | - | 7.49 | pIC50 | 32 | nM | IC50 | J Pharmacol Exp Ther (2014) 351: 538-48 [PMID:25253883] |
| tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597] | ||||||||
| GtoPdb | - | - | 9.3 | pIC50 | 0.5 | nM | IC50 | J Pharmacol Exp Ther (2014) 351: 538-48 [PMID:25253883] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
