AZD5069 [Ligand Id: 8948] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • CXCR1 in Human [GtoPdb: 68] [UniProtKB: P25024]
There should be some charts here, you may need to enable JavaScript!
  • CXCR2 in Human [GtoPdb: 69] [UniProtKB: P25025]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CXCR1 in Human [GtoPdb: 68] [UniProtKB: P25024]
GtoPdb Measuring displacement of CXCL8 binding to recombinant CXCR1 in HEK cell membrane preparations. - 6.9 pIC50 125 nM IC50 J. Pharmacol. Exp. Ther. (2015) 353: 340-50 [PMID:25736418]
CXCR2 in Human [GtoPdb: 69] [UniProtKB: P25025]
GtoPdb Measuring displacement of CXCL8 binding to recombinant CXCR2 in HEK cell membrane preparations. - 9.1 pIC50 0.79 nM IC50 J. Pharmacol. Exp. Ther. (2015) 353: 340-50 [PMID:25736418]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.