AZD5069 [Ligand Id: 8948] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CXCR1 in Human [GtoPdb: 68] [UniProtKB: P25024] | ||||||||
| GtoPdb | Measuring displacement of CXCL8 binding to recombinant CXCR1 in HEK cell membrane preparations. | - | 6.9 | pIC50 | 125 | nM | IC50 | J Pharmacol Exp Ther (2015) 353: 340-50 [PMID:25736418] |
| CXCR2 in Human [GtoPdb: 69] [UniProtKB: P25025] | ||||||||
| GtoPdb | Measuring displacement of CXCL8 binding to recombinant CXCR2 in HEK cell membrane preparations. | - | 9.1 | pIC50 | 0.79 | nM | IC50 | J Pharmacol Exp Ther (2015) 353: 340-50 [PMID:25736418] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
