FRAX486 [Ligand Id: 8938] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| p21 (RAC1) activated kinase 1 in Human [GtoPdb: 2133] [UniProtKB: Q13153] | ||||||||
| GtoPdb | - | - | 8.08 | pIC50 | 8.25 | nM | IC50 | Proc Natl Acad Sci USA (2013) 110: 5671-6 [PMID:23509247] |
| p21 (RAC1) activated kinase 2 in Human [GtoPdb: 2134] [UniProtKB: Q13177] | ||||||||
| GtoPdb | - | - | 7.4 | pIC50 | 39.5 | nM | IC50 | Proc Natl Acad Sci USA (2013) 110: 5671-6 [PMID:23509247] |
| p21 (RAC1) activated kinase 3 in Human [GtoPdb: 2135] [UniProtKB: O75914] | ||||||||
| GtoPdb | - | - | 7.26 | pIC50 | 55.3 | nM | IC50 | Proc Natl Acad Sci USA (2013) 110: 5671-6 [PMID:23509247] |
| p21 (RAC1) activated kinase 4 in Human [GtoPdb: 2136] [UniProtKB: O96013] | ||||||||
| GtoPdb | - | - | 6.11 | pIC50 | 779 | nM | IC50 | Proc Natl Acad Sci USA (2013) 110: 5671-6 [PMID:23509247] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
