liquiritigenin [Ligand Id: 8899] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL271939
  • TRPM3 in Human [GtoPdb: 495] [UniProtKB: Q9HCF6]
  • This target only has 0 pki data point
1 CHEMBL271939_lig_chart_1 TRPM3 Human
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  • Estrogen receptor-β in Human [GtoPdb: 621] [UniProtKB: Q92731]
  • This target only has 0 pki data point
2 CHEMBL271939_lig_chart_2 Estrogen receptor-β Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPM3 in Human [GtoPdb: 495] [UniProtKB: Q9HCF6]
GtoPdb - - 5.2 pIC50 - - - Mol. Pharmacol. (2013) 84: 736-50 [PMID:24006495]
Estrogen receptor-β in Human [GtoPdb: 621] [UniProtKB: Q92731]
GtoPdb Measuring activation of the ERE tk-Luc reporter by ER&bets; in transfected U2OS cells. - 7.44 pEC50 36.5 nM EC50 Mol. Cell. Endocrinol. (2008) 283: 49-57 [PMID:18177995]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]