liquiritigenin [Ligand Id: 8899] activity data from GtoPdb and ChEMBL

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

ChEMBL ligand: CHEMBL271939
  • TRPM3 in Human [GtoPdb: 495] [UniProtKB: Q9HCF6]
  • This target only has 0 pki data point
1 CHEMBL271939_lig_chart_1 TRPM3 Human
There should be some charts here, you may need to enable JavaScript!
  • Estrogen receptor-β in Human [GtoPdb: 621] [UniProtKB: Q92731]
  • This target only has 0 pki data point
2 CHEMBL271939_lig_chart_2 Estrogen receptor-β Human
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPM3 in Human [GtoPdb: 495] [UniProtKB: Q9HCF6]
GtoPdb - - 5.2 pIC50 - - - Mol. Pharmacol. (2013) 84: 736-50 [PMID:24006495]
Estrogen receptor-β in Human [GtoPdb: 621] [UniProtKB: Q92731]
GtoPdb Measuring activation of the ERE tk-Luc reporter by ER&bets; in transfected U2OS cells. - 7.44 pEC50 36.5 nM EC50 Mol. Cell. Endocrinol. (2008) 283: 49-57 [PMID:18177995]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]