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ChEMBL ligand: CHEMBL271939 |
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CHEMBL271939_lig_chart_1
TRPM3
Human
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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TRPM3 in Human [GtoPdb: 495] [UniProtKB: Q9HCF6] | ||||||||
GtoPdb | - | - | 5.2 | pIC50 | - | - | - | Mol. Pharmacol. (2013) 84: 736-50 [PMID:24006495] |
Estrogen receptor-β in Human [GtoPdb: 621] [UniProtKB: Q92731] | ||||||||
GtoPdb | Measuring activation of the ERE tk-Luc reporter by ER&bets; in transfected U2OS cells. | - | 7.44 | pEC50 | 36.5 | nM | EC50 | Mol. Cell. Endocrinol. (2008) 283: 49-57 [PMID:18177995] |
ChEMBL data shown on this page come from version 27:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]