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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143] | ||||||||
GtoPdb | Radioligand binding assay | - | 7.71 | pKi | 19.6 | nM | Ki |
NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407]; Life Sci (2003) 73: 663-678 [PMID:12801588] |
κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145] | ||||||||
GtoPdb | Radioligand binding assay | - | 8.94 | pKi | 1.14 | nM | Ki |
NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407]; ACS Chem Neurosci (2015) 6: 646-57 [PMID:25635572] |
μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372] | ||||||||
GtoPdb | Radioligand binding assay | - | 8.78 | pKi | 1.67 | nM | Ki |
NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407]; ACS Chem Neurosci (2015) 6: 646-57 [PMID:25635572] |
NOP receptor in Human [GtoPdb: 320] [UniProtKB: P41146] | ||||||||
GtoPdb | Radioligand binding assay | - | 8.76 | pKi | 1.75 | nM | Ki | ACS Chem Neurosci (2015) 6: 646-57 [PMID:25635572] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.