T-0632 [Ligand Id: 884] activity data from GtoPdb

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  • CCK1 receptor in Rat [GtoPdb: 76] [UniProtKB: P30551]
Created with Highcharts 10.3.3ValuesChart context menuCCK1 receptorpKd RatpKi RatpIC50 RatpEC50 Rat024681012Highcharts.com
  • GLP-1 receptor in Human [GtoPdb: 249] [UniProtKB: P43220]
Created with Highcharts 10.3.3ValuesChart context menuGLP-1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human012345Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CCK1 receptor in Rat [GtoPdb: 76] [UniProtKB: P30551]
GtoPdb - - 9.6 pIC50 0.25 nM IC50 Eur J Pharmacol (1996) 304: 147-54 [PMID:8813597]
GLP-1 receptor in Human [GtoPdb: 249] [UniProtKB: P43220]
GtoPdb - - 4.7 pIC50 21000 nM IC50 J Biol Chem (2001) 276: 37787-93 [PMID:11498540]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.