CTA091 [Ligand Id: 8819] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL1627233 |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| CYP24A1 in Human [GtoPdb: 1365] [UniProtKB: Q07973] | ||||||||
| GtoPdb | - | - | 8.2 | pIC50 | - | - | - | J Steroid Biochem Mol Biol (2010) 121: 13-9 [PMID:20347976] |
| CYP27A1 in Human [GtoPdb: 1369] [UniProtKB: Q02318] | ||||||||
| GtoPdb | - | - | 6 | pIC50 | >1000 | nM | IC50 | J Med Chem (2004) 47: 6854-63 [PMID:15615534] |
| CYP27B1 in Human [GtoPdb: 1370] [UniProtKB: O15528] | ||||||||
| GtoPdb | - | - | 6.26 | pIC50 | 554 | nM | IC50 | J Med Chem (2004) 47: 6854-63 [PMID:15615534] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
