TM38837 [Ligand Id: 8705] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CB1 receptor in Human [GtoPdb: 56] [UniProtKB: P21554] | ||||||||
| GtoPdb | Determined in a GTPγS assay | - | 7.62 | pIC50 | 24 | nM | IC50 | Bioorg Med Chem Lett (2024) 98: 129572 [PMID:38043690] |
| GtoPdb | Determined as antagonism in a GTPγS assay. | - | 8.07 | pIC50 | 6.7 | nM | IC50 |
ChemMedChem (2010) 5: 1439-43 [PMID:20652930]; Bioorg Med Chem Lett (2024) 98: 129572 [PMID:38043690] |
| CB2 receptor in Human [GtoPdb: 57] [UniProtKB: P34972] | ||||||||
| GtoPdb | - | - | 6.22 | pIC50 | 605 | nM | IC50 | ChemMedChem (2010) 5: 1439-43 [PMID:20652930] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
