PFI-4 [Ligand Id: 8575] activity data from GtoPdb

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  • bromodomain and PHD finger containing 1 in Human [GtoPdb: 2730] [UniProtKB: P55201]
Created with Highcharts 10.3.3ValuesChart context menubromodomain and PHD finger containing 1pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
bromodomain and PHD finger containing 1 in Human [GtoPdb: 2730] [UniProtKB: P55201]
GtoPdb Isothermal titration calorimetry (ITC) assay measuring binding to the BRPF1B isoform. - 7.89 pKd 13 nM Kd PFI-4 A chemical probe for BRPF1B.. thesgc.org

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.