chaetocin [Ligand Id: 8388] activity data from GtoPdb

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  • SUV39H1 histone lysine methyltransferase in Human [GtoPdb: 2715] [UniProtKB: O43463]
Created with Highcharts 10.3.3ValuesChart context menuSUV39H1 histone lysine methyltransferasepKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
SUV39H1 histone lysine methyltransferase in Human [GtoPdb: 2715] [UniProtKB: O43463]
GtoPdb - - 6.96 pIC50 110 nM IC50 Nat Chem Biol (2005) 1: 143-5 [PMID:16408017];
Nat Chem Biol (2013) 9: 136-7 [PMID:23416387]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.