LB42908 [Ligand Id: 8028] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| farnesyltransferase, CAAX box, subunit beta in Human [GtoPdb: 2826] [UniProtKB: P49356] | ||||||||
| GtoPdb | Measured as inhibition of FTase transfer of [3H]-farnesylpyrophosphate (FPP) to HRAS (0.9nM) or NRAS (2.4nM) | - | 9.05 | pIC50 | 0.9 | nM | IC50 | Bioorg Med Chem Lett (2001) 11: 3069-72 [PMID:11714612] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
