BrP-LPA [Ligand Id: 6985] activity data from GtoPdb

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  • LPA1 receptor in Human [GtoPdb: 272] [UniProtKB: Q92633]
Created with Highcharts 10.3.3ValuesChart context menuLPA1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human01234567Highcharts.com
  • LPA2 receptor in Mouse [GtoPdb: 273] [UniProtKB: Q9JL06]
Created with Highcharts 10.3.3ValuesChart context menuLPA2 receptorpKd MousepKi MousepIC50 MousepEC50 Mouse02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
LPA1 receptor in Human [GtoPdb: 272] [UniProtKB: Q92633]
GtoPdb - - 6.09 pKi 805 nM Ki Cancer Res (2009) 69: 5441-9 [PMID:19509223]
GtoPdb - - 5.34 pIC50 4520 nM IC50 Cancer Res (2009) 69: 5441-9 [PMID:19509223]
LPA2 receptor in Mouse [GtoPdb: 273] [UniProtKB: Q9JL06]
GtoPdb - - 6.61 pKi 245 nM Ki Cancer Res (2009) 69: 5441-9 [PMID:19509223]
GtoPdb - - 6.33 pIC50 468 nM IC50 Cancer Res (2009) 69: 5441-9 [PMID:19509223]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.