D-Nal-Cys-Tyr-D-Trp-Lys-Val-Cys-Nal-NH2 [Ligand Id: 635] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| BB1 receptor in Human [GtoPdb: 38] [UniProtKB: P28336] | ||||||||
| GtoPdb | - | - | 6.56 | pIC50 | 275 | nM | IC50 | Peptides (2009) 30: 1473-86 [PMID:19463875] |
| BB1 receptor in Rat [GtoPdb: 38] [UniProtKB: P24053] | ||||||||
| GtoPdb | - | - | 7.23 | pKi | 59 | nM | Ki | J Pharmacol Exp Ther (1999) 290: 1202-11 [PMID:10454496] |
| GtoPdb | - | - | 6 | pIC50 | 997 | nM | IC50 | Mol Pharmacol (1993) 44: 841-50 [PMID:7901752] |
| BB2 receptor in Human [GtoPdb: 39] [UniProtKB: P30550] | ||||||||
| GtoPdb | - | - | 6.77 | pKi | 170 | nM | Ki | J Pharmacol Exp Ther (1999) 290: 1202-11 [PMID:10454496] |
| GtoPdb | - | - | 5.61 | pIC50 | 2460 | nM | IC50 | Peptides (2009) 30: 1473-86 [PMID:19463875] |
| GtoPdb | - | - | 5.61 | pIC50 | 2460 | nM | IC50 | Peptides (2009) 30: 1473-86 [PMID:19463875] |
| BB2 receptor in Rat [GtoPdb: 39] [UniProtKB: P52500] | ||||||||
| GtoPdb | - | - | 5 | pKi | >10000 | nM | Ki | Biochemistry (1999) 38: 7307-20 [PMID:10353842] |
| BB3 receptor in Human [GtoPdb: 40] [UniProtKB: P32247] | ||||||||
| GtoPdb | - | - | 5.6 | pIC50 | - | - | - |
J Biol Chem (1997) 272: 26062-71 [PMID:9325344]; J Pharmacol Exp Ther (1998) 287: 366-80 [PMID:9765358]; J Biol Chem (1998) 273: 13613-24 [PMID:9593699] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
