galanin(2-29) (pig) [Ligand Id: 6130] activity data from GtoPdb

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  • GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211]
  • GAL1 receptor in Rat [GtoPdb: 243] [UniProtKB: Q62805]
Created with Highcharts 10.3.3ValuesChart context menuGAL1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
  • GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603]
Created with Highcharts 10.3.3ValuesChart context menuGAL2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755]
Created with Highcharts 10.3.3ValuesChart context menuGAL3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211]
GtoPdb - - 7.58 pKi 26.3 nM Ki Peptides (1998) 19: 1771-81 [PMID:9880084]
GtoPdb - - 7.52 pIC50 30.4 nM IC50 Brain Res Mol Brain Res (1998) 58: 156-69 [PMID:9685625]
GAL1 receptor in Rat [GtoPdb: 243] [UniProtKB: Q62805]
GtoPdb - - 8.15 pKi 7.14 nM Ki Brain Res Mol Brain Res (1995) 34: 179-89 [PMID:8750821];
J Mol Neurosci (1995) 6: 33-41 [PMID:8562318]
GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603]
GtoPdb - - 8.54 pKi 2.88 nM Ki Peptides (1998) 19: 1771-81 [PMID:9880084]
GtoPdb - - 8.74 pIC50 1.8 nM IC50 Brain Res Mol Brain Res (1997) 51: 49-59 [PMID:9427506];
Brain Res Mol Brain Res (1998) 58: 156-69 [PMID:9685625]
GtoPdb - - 8.93 pEC50 1.17 nM EC50 Peptides (1998) 19: 1771-81 [PMID:9880084];
Brain Res Mol Brain Res (1998) 58: 156-69 [PMID:9685625]
GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755]
GtoPdb - - 7.22 pKi 60.26 nM Ki Peptides (1998) 19: 1771-81 [PMID:9880084]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.