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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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BB1 receptor in Human [GtoPdb: 38] [UniProtKB: P28336] | ||||||||
GtoPdb | - | - | 10.3 | pKi | 0.05 | nM | Ki |
Pharmacol Rev (2008) 60: 1-42 [PMID:18055507]; Peptides (2011) 32: 1685-99 [PMID:21729729]; Peptides (2015) 72: 128-44 [PMID:25976083] |
BB2 receptor in Human [GtoPdb: 39] [UniProtKB: P30550] | ||||||||
GtoPdb | - | - | 8.13 | pKi | 7.4 | nM | Ki |
J Pharmacol Exp Ther (1999) 290: 1202-11 [PMID:10454496]; Mol Pharmacol (1995) 47: 10-20 [PMID:7838118] |
GtoPdb | - | - | 7.52 | pIC50 | 30.1 | nM | IC50 |
Peptides (2011) 32: 1685-99 [PMID:21729729]; Peptides (2009) 30: 1473-86 [PMID:19463875] |
BB2 receptor in Mouse [GtoPdb: 39] [UniProtKB: P21729] | ||||||||
GtoPdb | - | - | 7.38 | pKi | 42 | nM | Ki | Mol Pharmacol (1995) 47: 10-20 [PMID:7838118] |
BB2 receptor in Rat [GtoPdb: 39] [UniProtKB: P52500] | ||||||||
GtoPdb | - | - | 6.61 | pKi | 248 | nM | Ki | J Pharmacol Exp Ther (1999) 290: 1202-11 [PMID:10454496] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.