galanin(D-Trp2) (pig) [Ligand Id: 6095] activity data from GtoPdb

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  • GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211]
  • GAL1 receptor in Rat [GtoPdb: 243] [UniProtKB: Q62805]
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  • GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603]
  • GAL2 receptor in Rat [GtoPdb: 244] [UniProtKB: O08726]
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  • GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755]
  • GAL3 receptor in Rat [GtoPdb: 245] [UniProtKB: O88626]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211]
GtoPdb - - 6.2 pKi 630.96 nM Ki Peptides (1998) 19: 1771-81 [PMID:9880084]
GAL1 receptor in Rat [GtoPdb: 243] [UniProtKB: Q62805]
GtoPdb - - 6.39 pKi 407.4 nM Ki J Biol Chem (1997) 272: 24612-6 [PMID:9305929];
J Biol Chem (1998) 273: 23321-6 [PMID:9722565]
GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603]
GtoPdb - - 6.7 pKi 199.53 nM Ki Peptides (1998) 19: 1771-81 [PMID:9880084]
GtoPdb - - 6.47 pEC50 338.84 nM EC50 Peptides (1998) 19: 1771-81 [PMID:9880084]
GAL2 receptor in Rat [GtoPdb: 244] [UniProtKB: O08726]
GtoPdb - - 8.15 pKi 7 nM Ki J Biol Chem (1997) 272: 24612-6 [PMID:9305929];
J Biol Chem (1998) 273: 23321-6 [PMID:9722565]
GtoPdb - - 6.82 pEC50 150 nM EC50 J Biol Chem (1997) 272: 24612-6 [PMID:9305929]
GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755]
GtoPdb - - 6 pKi >1000 nM Ki J Biol Chem (1998) 273: 23321-6 [PMID:9722565]
GAL3 receptor in Rat [GtoPdb: 245] [UniProtKB: O88626]
GtoPdb - - 6 pKi >1000 nM Ki J Biol Chem (1998) 273: 23321-6 [PMID:9722565];
Peptides (1998) 19: 1771-81 [PMID:9880084]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.