p38 MAP kinase inhibitor [Ligand Id: 6013] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL91730 |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| mitogen-activated protein kinase 14/MAP kinase p38 alpha in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4825] [GtoPdb: 1499] [UniProtKB: P70618] | ||||||||
| ChEMBL | Inhibitory potency evaluated against rat p38 kinase | B | 7.46 | pIC50 | 35 | nM | IC50 | Bioorg. Med. Chem. Lett. (1998) 8: 2689-2694 [PMID:9873604] |
ChEMBL data shown on this page come from version 31:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]
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