p38 MAP kinase inhibitor [Ligand Id: 6013] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL91730
  • mitogen-activated protein kinase 14/MAP kinase p38 alpha in Rat [ChEMBL: CHEMBL4825] [GtoPdb: 1499] [UniProtKB: P70618]
  • This target only has 0 pki data point
  • 0
1 CHEMBL91730_lig_chart_1 MAP kinase p38 alpha Rat
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
mitogen-activated protein kinase 14/MAP kinase p38 alpha in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4825] [GtoPdb: 1499] [UniProtKB: P70618]
ChEMBL Inhibitory potency evaluated against rat p38 kinase B 7.46 pIC50 35 nM IC50 Bioorg. Med. Chem. Lett. (1998) 8: 2689-2694 [PMID:9873604]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]