ChEMBL ligand: CHEMBL2178734
cyclin dependent kinase 1 in Human [GtoPdb: 1961] [UniProtKB: P06493] There should be some charts here, you may need to enable JavaScript!
cyclin dependent kinase 5 in Human [GtoPdb: 1977] [UniProtKB: Q00535] There should be some charts here, you may need to enable JavaScript!
glycogen synthase kinase 3 alpha in Pig [GtoPdb: 2029] There should be some charts here, you may need to enable JavaScript!
glycogen synthase kinase 3 beta in Pig [GtoPdb: 2030] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
cyclin dependent kinase 1 in Human [GtoPdb: 1961] [UniProtKB: P06493]
GtoPdb	CDK1/cyclin B complex	-	6.49	pIC50	320	nM	IC50	J Med Chem (2004) 47: 935-46 [PMID:14761195]; Chem Biol (2003) 10: 1255-66 [PMID:14700633]
cyclin dependent kinase 5 in Human [GtoPdb: 1977] [UniProtKB: Q00535]
GtoPdb	CDK5/p25 complex	-	7.08	pIC50	83	nM	IC50	J Med Chem (2004) 47: 935-46 [PMID:14761195]; Chem Biol (2003) 10: 1255-66 [PMID:14700633]
glycogen synthase kinase 3 alpha in Pig [GtoPdb: 2029]
GtoPdb	GSK3α/β complex from pig brain	-	8.3	pIC50	5	nM	IC50	J Med Chem (2004) 47: 935-46 [PMID:14761195]; Chem Biol (2003) 10: 1255-66 [PMID:14700633]
glycogen synthase kinase 3 beta in Pig [GtoPdb: 2030]
GtoPdb	GSK3α/β complex from pig brain	-	8.3	pIC50	5	nM	IC50	J Med Chem (2004) 47: 935-46 [PMID:14761195]; Chem Biol (2003) 10: 1255-66 [PMID:14700633]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]