2-phenyl-propylamine [Ligand Id: 5510] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL158578 (2-Phenyl-Propylamine)
  • TA1 receptor in Human [GtoPdb: 364] [UniProtKB: Q96RJ0]
Created with Highcharts 10.3.3ValuesChart context menuTA1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TA1 receptor in Human [GtoPdb: 364] [UniProtKB: Q96RJ0]
GtoPdb - - 6.98 pEC50 104 nM EC50 J Pharmacol Exp Ther (2007) 320: 475-85 [PMID:17038507]

ChEMBL data shown on this page come from version 35:

Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]