ChEMBL ligand: CHEMBL117785 (Nitoman, NSC-169886, Revocon, RO 1-9569, RO-1-9569, RO-19569, Tetmodis, Tetrabenazine, Xenazine, Xenazine 25)
Vesicular monoamine transporter 2 in Human [GtoPdb: 1012] [UniProtKB: Q05940] Synaptic vesicular amine transporter in Bovine [ChEMBL: CHEMBL4271] [UniProtKB: Q27963] Vesicular monoamine transporter 2/Synaptic vesicular amine transporter in Rat [ChEMBL: CHEMBL4828] [GtoPdb: 1012] [UniProtKB: Q01827] There should be some charts here, you may need to enable JavaScript!
Vesicular monoamine transporter 1 in Human [GtoPdb: 1011] [UniProtKB: P54219] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
Vesicular monoamine transporter 2 in Human [GtoPdb: 1012] [UniProtKB: Q05940]
GtoPdb	-	-	7	pKi	97	nM	Ki	Proc Natl Acad Sci USA (1996) 93: 5166-71 [PMID:8643547]
Synaptic vesicular amine transporter in Bovine (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4271] [UniProtKB: Q27963]
ChEMBL	Inhibition of dopamine uptake at VMAT in bovine chromaffin granule ghosts	B	8.4	pKi	4	nM	Ki	J Med Chem (2008) 51: 760-768 [PMID:18220329]
Vesicular monoamine transporter 2/Synaptic vesicular amine transporter in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4828] [GtoPdb: 1012] [UniProtKB: Q01827]
ChEMBL	Inhibition of [3H]dopamine uptake at VMAT2 in rat brain synaptic vesicle by liquid scintillation spectroscopy	B	7.27	pKi	54	nM	Ki	J Med Chem (2009) 52: 7878-7882 [PMID:19691331]
ChEMBL	Displacement of [3H]DTBZ from VMAT2 dihydrotetrabenazine binding site in rat brain synaptic vesicle by scintillation counting	B	7.89	pKi	13	nM	Ki	J Med Chem (2009) 52: 7878-7882 [PMID:19691331]
ChEMBL	Displacement of [3H]MTBZ from VMAT2 in rat whole brain vesicles by liquid scintillation spectrophotometry	B	7.89	pKi	13	nM	Ki	Bioorg Med Chem (2010) 18: 640-649 [PMID:20036131]
ChEMBL	Displacement of [3H]DHTBZ from Sprague-Dawley rat striatum VMAT2 after 1 hr by liquid scintillation counting	B	8.12	pKi	7.62	nM	Ki	Eur J Med Chem (2011) 46: 1841-1848 [PMID:21396745]
Vesicular monoamine transporter 1 in Human [GtoPdb: 1011] [UniProtKB: P54219]
GtoPdb	-	-	4.7	pKi	20000	nM	Ki	Proc Natl Acad Sci USA (1996) 93: 5166-71 [PMID:8643547]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]