R3(BΔ23-27)R/I5 chimeric peptide [Ligand Id: 3907] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| RXFP3 in Human [GtoPdb: 353] [UniProtKB: Q9NSD7] | ||||||||
| GtoPdb | - | - | 8.49 | pKi | - | - | - | J Am Chem Soc (2011) 133: 4965-74 [PMID:21384867] |
| GtoPdb | - | - | 8.1 | pIC50 | - | - | - | Eur J Pharmacol (2015) 747: 123-31 [PMID:25496752] |
| GtoPdb | - | - | 9.2 | pIC50 | 0.67 | nM | IC50 | J Biol Chem (2007) 282: 25425-35 [PMID:17606621] |
| GtoPdb | - | - | 9.4 | pIC50 | - | - | - | Eur J Pharmacol (2015) 747: 123-31 [PMID:25496752] |
| GtoPdb | - | - | 9.02 | pEC50 | - | - | - | Br J Pharmacol (2014) 171: 2827-41 [PMID:24641548] |
| RXFP3 in Rat [GtoPdb: 353] [UniProtKB: Q5Y986] | ||||||||
| GtoPdb | - | - | 9.2 | pIC50 | - | - | - | Eur J Pharmacol (2015) 747: 123-31 [PMID:25496752] |
| GtoPdb | - | - | 10.1 | pIC50 | - | - | - | Eur J Pharmacol (2015) 747: 123-31 [PMID:25496752] |
| RXFP4 in Human [GtoPdb: 354] [UniProtKB: Q8TDU9] | ||||||||
| GtoPdb | - | - | 8.64 | pIC50 | - | - | IC50 |
J Biol Chem (2007) 282: 25425-35 [PMID:17606621]; J Am Chem Soc (2011) 133: 4965-74 [PMID:21384867] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
