galanin(2-29) (rat/mouse) [Ligand Id: 3876] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211] | ||||||||
| GtoPdb | - | - | 8 | pIC50 | 10 | nM | IC50 | Biochem Biophys Res Commun (1997) 233: 823-8 [PMID:9168941] |
| GAL1 receptor in Mouse [GtoPdb: 243] [UniProtKB: P56479] | ||||||||
| GtoPdb | - | - | 7.97 | pKi | 10.8 | nM | Ki |
FEBS Lett (1997) 411: 225-30 [PMID:9271210]; J Neurochem (1998) 71: 2252-9 [PMID:9832122] |
| GAL1 receptor in Rat [GtoPdb: 243] [UniProtKB: Q62805] | ||||||||
| GtoPdb | - | - | 7.07 | pKi | 85 | nM | Ki |
Mol Pharmacol (1997) 52: 337-43 [PMID:9281594]; J Biol Chem (1997) 272: 31949-52 [PMID:9405385]; FEBS Lett (1998) 434: 277-82 [PMID:9742938] |
| GtoPdb | - | - | 8.14 | pIC50 | 7.2 | nM | IC50 |
Biochem Biophys Res Commun (1997) 233: 823-8 [PMID:9168941]; FEBS Lett (1997) 405: 285-90 [PMID:9108306] |
| GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603] | ||||||||
| GtoPdb | - | - | 9.04 | pKi | 0.91 | nM | Ki | Biochem Biophys Res Commun (1998) 243: 474-9 [PMID:9480833] |
| GAL2 receptor in Mouse [GtoPdb: 244] [UniProtKB: O88854] | ||||||||
| GtoPdb | - | - | 8.17 | pKi | 6.8 | nM | Ki | J Neurochem (1998) 71: 2252-9 [PMID:9832122] |
| GAL2 receptor in Rat [GtoPdb: 244] [UniProtKB: O08726] | ||||||||
| GtoPdb | - | - | 8.72 | pKi | 1.9 | nM | Ki |
Mol Pharmacol (1997) 52: 337-43 [PMID:9281594]; J Biol Chem (1997) 272: 31949-52 [PMID:9405385]; FEBS Lett (1998) 434: 277-82 [PMID:9742938]; J Neurochem (1998) 71: 2252-9 [PMID:9832122] |
| GtoPdb | - | - | 8.54 | pIC50 | 2.9 | nM | IC50 | FEBS Lett (1997) 405: 285-90 [PMID:9108306] |
| GAL3 receptor in Rat [GtoPdb: 245] [UniProtKB: O88626] | ||||||||
| GtoPdb | - | - | 7.9 | pKi | 12.6 | nM | Ki |
J Biol Chem (1997) 272: 31949-52 [PMID:9405385]; FEBS Lett (1998) 434: 277-82 [PMID:9742938] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
