[3H]5-CT [Ligand Id: 262] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1628596
  • 5-HT1D receptor in Human [GtoPdb: 3] [UniProtKB: P28221]
  • This target only has 0 pki data point
  • 0
1 CHEMBL1628596_lig_chart_1 5-HT1D receptor Human
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  • 5-HT5A receptor in Human [GtoPdb: 10] [UniProtKB: P47898]
  • This target only has 0 pki data point
  • 0
2 CHEMBL1628596_lig_chart_2 5-HT5A receptor Human
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  • 5-HT7 receptor in Human [GtoPdb: 12] [UniProtKB: P34969]
  • This target only has 0 pki data point
  • 0
3 CHEMBL1628596_lig_chart_3 5-HT7 receptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
5-HT1D receptor in Human [GtoPdb: 3] [UniProtKB: P28221]
GtoPdb - - 9.1 pKd 0.9 nM Kd FEBS Lett (1999) 456: 63-7 [PMID:10452531]
5-HT5A receptor in Human [GtoPdb: 10] [UniProtKB: P47898]
GtoPdb - - 8.6 pKd 2.5 nM Kd Eur J Pharmacol (2001) 418: 157-67 [PMID:11343685]
5-HT7 receptor in Human [GtoPdb: 12] [UniProtKB: P34969]
GtoPdb - - 9.4 pKd 0.4 nM Kd Br J Pharmacol (2000) 130: 409-17 [PMID:10807680]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]