tertiapin-Q [Ligand Id: 2383] activity data from GtoPdb

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  • Kir1.1 in Human [GtoPdb: 429] [UniProtKB: P48048]
  • Kir1.1 in Rat [GtoPdb: 429] [UniProtKB: P35560]
Created with Highcharts 10.3.3ValuesChart context menuKir1.1pKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
  • Kir3.1 in Rat [GtoPdb: 434] [UniProtKB: P63251]
Created with Highcharts 10.3.3ValuesChart context menuKir3.1pKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
  • Kir3.4 in Rat [GtoPdb: 437] [UniProtKB: P48548]
Created with Highcharts 10.3.3ValuesChart context menuKir3.4pKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Kir1.1 in Human [GtoPdb: 429] [UniProtKB: P48048]
GtoPdb - - 8.9 pIC50 - - - Biochemistry (1999) 38: 14286-93 [PMID:10572003]
Kir1.1 in Rat [GtoPdb: 429] [UniProtKB: P35560]
GtoPdb - - 8.7 pKi - - - Biochemistry (1999) 38: 14286-93 [PMID:10572003]
GtoPdb - - 8.9 pKi - - - Biochemistry (2006) 45: 10129-39 [PMID:16906771];
Biochemistry (1999) 38: 14286-93 [PMID:10572003]
Kir3.1 in Rat [GtoPdb: 434] [UniProtKB: P63251]
GtoPdb - - 8 pEC50 10 nM EC50 Biochemistry (1998) 37: 13291-9 [PMID:9748337]
Kir3.4 in Rat [GtoPdb: 437] [UniProtKB: P48548]
GtoPdb - - 8.1 pKi - - - Biochemistry (1998) 37: 13291-9 [PMID:9748337]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.