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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| KCa2.1 in Human [GtoPdb: 381] [UniProtKB: Q92952] | ||||||||
| GtoPdb | - | - | 7.1 | pIC50 | 80 | nM | IC50 |
Br J Pharmacol (2000) 129: 991-9 [PMID:10696100]; J Biol Chem (2001) 276: 43145-51 [PMID:11527975] |
| KCa2.2 in Human [GtoPdb: 382] [UniProtKB: Q9H2S1] | ||||||||
| GtoPdb | - | - | 9.7 | pIC50 | - | - | - |
J Biol Chem (2001) 276: 43145-51 [PMID:11527975]; FEBS Lett (2000) 469: 196-202 [PMID:10713270] |
| KCa2.2 in Rat [GtoPdb: 382] [UniProtKB: P70604] | ||||||||
| GtoPdb | - | - | 9.5 | pIC50 | - | - | - | Br J Pharmacol (2000) 129: 991-9 [PMID:10696100] |
| KCa2.3 in Human [GtoPdb: 383] [UniProtKB: Q9UGI6] | ||||||||
| GtoPdb | - | - | 9 | pIC50 | - | - | - |
J Biol Chem (2001) 276: 43145-51 [PMID:11527975]; Mol Pharmacol (2004) 65: 788-801 [PMID:14978258] |
| KCa2.3 in Rat [GtoPdb: 383] [UniProtKB: P70605] | ||||||||
| GtoPdb | - | - | 8.1 | pIC50 | - | - | - | J Physiol (Lond.) (2001) 535: 323-34 [PMID:11533126] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.