d[Cha4]LVP [Ligand Id: 2188] activity data from GtoPdb

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  • V1A receptor in Rat [GtoPdb: 366] [UniProtKB: P30560]
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  • V1B receptor in Rat [GtoPdb: 367] [UniProtKB: P48974]
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  • V2 receptor in Rat [GtoPdb: 368] [UniProtKB: Q00788]
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  • OT receptor in Rat [GtoPdb: 369] [UniProtKB: P70536]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
V1A receptor in Rat [GtoPdb: 366] [UniProtKB: P30560]
GtoPdb - - 5 pKi - - - J Med Chem (2007) 50: 835-847 [PMID:17300166]
V1B receptor in Rat [GtoPdb: 367] [UniProtKB: P48974]
GtoPdb - - 8.7 pKi - - - J Med Chem (2007) 50: 835-847 [PMID:17300166]
V2 receptor in Rat [GtoPdb: 368] [UniProtKB: Q00788]
GtoPdb - - 6.2 pKi - - - J Med Chem (2007) 50: 835-847 [PMID:17300166]
OT receptor in Rat [GtoPdb: 369] [UniProtKB: P70536]
GtoPdb - - 6.2 pKi - - - J Med Chem (2007) 50: 835-847 [PMID:17300166]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.