d[Cha4]AVP [Ligand Id: 2187] activity data from GtoPdb

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  • V1A receptor in Human [GtoPdb: 366] [UniProtKB: P37288]
Created with Highcharts 10.3.3ValuesChart context menuV1A receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • V1B receptor in Human [GtoPdb: 367] [UniProtKB: P47901]
Created with Highcharts 10.3.3ValuesChart context menuV1B receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
  • V2 receptor in Human [GtoPdb: 368] [UniProtKB: P30518]
Created with Highcharts 10.3.3ValuesChart context menuV2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • OT receptor in Human [GtoPdb: 369] [UniProtKB: P30559]
Created with Highcharts 10.3.3ValuesChart context menuOT receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
V1A receptor in Human [GtoPdb: 366] [UniProtKB: P37288]
GtoPdb - - 7.1 pKi - - - Endocrinology (2002) 143: 4655-64 [PMID:12446593]
V1B receptor in Human [GtoPdb: 367] [UniProtKB: P47901]
GtoPdb - - 9.7 pKi - - - Endocrinology (2002) 143: 4655-64 [PMID:12446593];
Br J Pharmacol (2005) 146: 744-751 [PMID:16158071]
V2 receptor in Human [GtoPdb: 368] [UniProtKB: P30518]
GtoPdb - - 6.5 pKi - - - Endocrinology (2002) 143: 4655-64 [PMID:12446593]
OT receptor in Human [GtoPdb: 369] [UniProtKB: P30559]
GtoPdb - - 7.7 pKi - - - Endocrinology (2002) 143: 4655-64 [PMID:12446593];
Br J Pharmacol (2005) 146: 744-751 [PMID:16158071]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.