BIM 23197 [Ligand Id: 2041] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
Created with Highcharts 10.3.3ValuesChart context menuSST2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
  • SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
Created with Highcharts 10.3.3ValuesChart context menuSST3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
Created with Highcharts 10.3.3ValuesChart context menuSST5 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
GtoPdb - - 9.7 pIC50 - - - J Clin Invest (1997) 99: 789-98 [PMID:9045884]
SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
GtoPdb - - 7.6 pIC50 - - - J Clin Invest (1997) 99: 789-98 [PMID:9045884]
SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
GtoPdb - - 8 pIC50 - - - J Clin Invest (1997) 99: 789-98 [PMID:9045884]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.