BIM 23023 [Ligand Id: 2032] activity data from GtoPdb

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  • SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
  • SST2 receptor in Mouse [GtoPdb: 356] [UniProtKB: P30875]
  • SST2 receptor in Rat [GtoPdb: 356] [UniProtKB: P30680]
Created with Highcharts 10.3.3ValuesChart context menuSST2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd MousepKi MousepIC50 MousepEC50 MousepKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
  • SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
  • SST3 receptor in Mouse [GtoPdb: 357] [UniProtKB: P30935]
  • SST3 receptor in Rat [GtoPdb: 357] [UniProtKB: P30936]
Created with Highcharts 10.3.3ValuesChart context menuSST3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd MousepKi MousepIC50 MousepEC50 MousepKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
  • SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
  • SST5 receptor in Rat [GtoPdb: 359] [UniProtKB: P30938]
Created with Highcharts 10.3.3ValuesChart context menuSST5 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
GtoPdb - - 9.4 pKi - - - Endocrinology (1994) 135: 2814-7 [PMID:7988476]
SST2 receptor in Mouse [GtoPdb: 356] [UniProtKB: P30875]
GtoPdb - - 9.4 pKi - - - Rev Physiol Biochem Pharmacol (1998) 133: 55-108 [PMID:9600011]
SST2 receptor in Rat [GtoPdb: 356] [UniProtKB: P30680]
GtoPdb - - 9.2 pKi - - - Rev Physiol Biochem Pharmacol (1998) 133: 55-108 [PMID:9600011]
SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
GtoPdb - - 8.1 pKi - - - Endocrinology (1994) 135: 2814-7 [PMID:7988476]
SST3 receptor in Mouse [GtoPdb: 357] [UniProtKB: P30935]
GtoPdb - - 7.9 pIC50 - - - Mol Pharmacol (1993) 43: 838-44 [PMID:8100350]
SST3 receptor in Rat [GtoPdb: 357] [UniProtKB: P30936]
GtoPdb - - 7 pKi - - - Rev Physiol Biochem Pharmacol (1998) 133: 55-108 [PMID:9600011]
SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
GtoPdb - - 9.4 pKi - - - Rev Physiol Biochem Pharmacol (1998) 133: 55-108 [PMID:9600011];
Endocrinology (1994) 135: 2814-7 [PMID:7988476]
SST5 receptor in Rat [GtoPdb: 359] [UniProtKB: P30938]
GtoPdb - - 7.8 pKi - - - Rev Physiol Biochem Pharmacol (1998) 133: 55-108 [PMID:9600011]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.