relaxin [Ligand Id: 1989] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| RXFP1 in Human [GtoPdb: 351] [UniProtKB: Q9HBX9] | ||||||||
| GtoPdb | - | - | 10.2 | pKi | - | - | - |
J Biol Chem (2003) 278: 7855-62 [PMID:12506116]; J Pharmacol Exp Ther (2005) 313: 677-87 [PMID:15649866]; J Biol Chem (2008) 283: 17287-97 [PMID:18434306] |
| GtoPdb | - | - | 10.37 | pEC50 | - | - | - | J Biol Chem (2008) 283: 17287-97 [PMID:18434306] |
| RXFP2 in Human [GtoPdb: 352] [UniProtKB: Q8WXD0] | ||||||||
| GtoPdb | - | - | 8.48 | pKi | - | - | - |
J Pharmacol Exp Ther (2005) 313: 677-87 [PMID:15649866]; J Biol Chem (2008) 283: 17287-97 [PMID:18434306] |
| GtoPdb | - | - | 9.13 | pEC50 | - | - | - | J Biol Chem (2008) 283: 17287-97 [PMID:18434306] |
| RXFP3 in Human [GtoPdb: 353] [UniProtKB: Q9NSD7] | ||||||||
| GtoPdb | - | - | 10 | pKd | - | - | - | Mol Pharmacol (2010) 77: 759-72 [PMID:20159943] |
| GtoPdb | - | - | 8.35 | pEC50 | - | - | - |
Mol Pharmacol (2010) 77: 759-72 [PMID:20159943]; Br J Pharmacol (2014) 171: 2827-41 [PMID:24641548] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
