S 16924 [Ligand Id: 167] activity data from GtoPdb

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  • 5-HT1A receptor in Human [GtoPdb: 1] [UniProtKB: P08908]
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  • 5-HT2A receptor in Human [GtoPdb: 6] [UniProtKB: P28223]
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  • 5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595]
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  • 5-HT2C receptor in Human [GtoPdb: 8] [UniProtKB: P28335]
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  • 5-HT6 receptor in Rat [GtoPdb: 11] [UniProtKB: P31388]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
5-HT1A receptor in Human [GtoPdb: 1] [UniProtKB: P08908]
GtoPdb - - 8.4 pKi - - - J Pharmacol Exp Ther (1998) 286: 1341-55 [PMID:9732398]
5-HT2A receptor in Human [GtoPdb: 6] [UniProtKB: P28223]
GtoPdb - - 9 pKi - - - J Pharmacol Exp Ther (1998) 286: 1341-55 [PMID:9732398]
5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595]
GtoPdb - - 8.4 pKi - - - J Pharmacol Exp Ther (1998) 286: 1341-55 [PMID:9732398]
5-HT2C receptor in Human [GtoPdb: 8] [UniProtKB: P28335]
GtoPdb - - 7.7 pKi - - - J Pharmacol Exp Ther (1998) 286: 1341-55 [PMID:9732398]
5-HT6 receptor in Rat [GtoPdb: 11] [UniProtKB: P31388]
GtoPdb - - 7.6 pKi - - - J Pharmacol Exp Ther (1998) 286: 1341-55 [PMID:9732398]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.