garutadustat [Ligand Id: 14465] activity data from GtoPdb

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  • egl-9 family hypoxia inducible factor 1 in Human [GtoPdb: 2833] [UniProtKB: Q9GZT9]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
egl-9 family hypoxia inducible factor 1 in Human [GtoPdb: 2833] [UniProtKB: Q9GZT9]
GtoPdb - - 8.3 pIC50 <5 nM IC50 WO2023072246A1. Prolyl hydroxylase domain-containing protein (phd) inhibitors and uses thereof (2023)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.