SGC-CK1γ-1 [Ligand Id: 14339] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| casein kinase 1 gamma 1 in Human [GtoPdb: 1999] [UniProtKB: Q9HCP0] | ||||||||
| GtoPdb | Determined in a NanoBRET assay | - | 6.74 | pIC50 | 180 | nM | IC50 | J Med Chem (2026) 69: 2666-2684 [PMID:41587072] |
| GtoPdb | Determined in an enzyme activity assay | - | 7.55 | pIC50 | 28 | nM | IC50 | J Med Chem (2026) 69: 2666-2684 [PMID:41587072] |
| casein kinase 1 gamma 2 in Human [GtoPdb: 2000] [UniProtKB: P78368] | ||||||||
| GtoPdb | Determined in a NanoBRET assay | - | 6.74 | pIC50 | 180 | nM | IC50 | J Med Chem (2026) 69: 2666-2684 [PMID:41587072] |
| GtoPdb | Determined in an enzyme activity assay | - | 8.15 | pIC50 | 7 | nM | IC50 | J Med Chem (2026) 69: 2666-2684 [PMID:41587072] |
| casein kinase 1 gamma 3 in Human [GtoPdb: 2001] [UniProtKB: Q9Y6M4] | ||||||||
| GtoPdb | Determined in an enzyme activity assay | - | 6.02 | pIC50 | 958 | nM | IC50 | J Med Chem (2026) 69: 2666-2684 [PMID:41587072] |
| GtoPdb | Determined in a NanoBRET assay | - | 6.64 | pIC50 | 230 | nM | IC50 | J Med Chem (2026) 69: 2666-2684 [PMID:41587072] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
