PF-07899895 [Ligand Id: 14208] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| salt inducible kinase 1 in Human [GtoPdb: 2197] [UniProtKB: P57059] | ||||||||
| GtoPdb | - | - | 8.92 | pIC50 | 1.2 | nM | IC50 | WO2024062360A1. Heterocyclic sik inhibitors (2024) |
| salt inducible kinase 2 in Human [GtoPdb: 2198] [UniProtKB: Q9H0K1] | ||||||||
| GtoPdb | - | - | 9.05 | pIC50 | 0.9 | nM | IC50 | WO2024062360A1. Heterocyclic sik inhibitors (2024) |
| SIK family kinase 3 in Human [GtoPdb: 2199] [UniProtKB: Q9Y2K2] | ||||||||
| GtoPdb | - | - | 8.74 | pIC50 | 1.8 | nM | IC50 | WO2024062360A1. Heterocyclic sik inhibitors (2024) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
