limertinib [Ligand Id: 14195] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| epidermal growth factor receptor in Human [GtoPdb: 1797] [UniProtKB: P00533] | ||||||||
| GtoPdb | Inhibition of WT EGFR | - | 8.22 | pIC50 | 6 | nM | IC50 | Mol Cancer (2020) 19: 90 [PMID:32404161] |
| GtoPdb | Inhibition of EGFRexon19del | - | 9.3 | pIC50 | 0.5 | nM | IC50 | Mol Cancer (2020) 19: 90 [PMID:32404161] |
| GtoPdb | Inhibition of EGFRT790M | - | 9.3 | pIC50 | 0.5 | nM | IC50 | Mol Cancer (2020) 19: 90 [PMID:32404161] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
